1rm8 A 1.8 BS01 ZN A 1 H246 H250 H256 H123 H127 H133 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 P51512 14741217 500 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP 1rm8 A 1.8 BS02 ZN A 2 H193 D195 H208 H221 H70 D72 H85 H98 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 P51512 14741217 501 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP 1rm8 A 1.8 BS03 CA A 1 D200 G201 G203 F205 D223 E226 D77 G78 G80 F82 D100 E103 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 P51512 14741217 502 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP 1rm8 A 1.8 BS04 CA A 2 D183 G215 I216 G217 D219 D60 G92 I93 G94 D96 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 P51512 14741217 504 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP 1rm8 A 1.8 BS05 BAT A 1 G204 F205 L206 A207 V243 H246 E247 H250 H256 P266 F267 Y268 G81 F82 L83 A84 V120 H123 E124 H127 H133 P143 F144 Y145 H246 E247 H250 H256 H123 E124 H127 H133 3.4.24.- 0004222,0006508,0008237,0008270,0031012 -logKd/Ki=9.00, Ki=1nM P51512 14741217 800 GQKWQHKHITYSIKNVTPKVGDPETRKAIRRAFDVWQNVTPLTFEEVPYSELENGKRDVDITIIFASGFHGDSSPFDGEGGFLAHAYFPGPGIGGDTHFDSDEPWTLGNPNHDGNDLFLVAVHELGHALGLEHSNDPTAIMAPFYQYMETDNFKLPNDDLQGIQKIYGP