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Structure of PDB 4mg7 Chain A Binding Site BS01

Receptor Information
>4mg7 Chain A (length=239) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
SLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADREL
VHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLF
APNLLLDRNQEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGV
YTFSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLI
LSHIRHMSNKGMEHLYSMKCKNVVPLSDLLLEMLDAHRL
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB4mg7 Structural and functional profiling of environmental ligands for estrogen receptors.
Resolution2.15 Å
Binding residue
(original residue number in PDB)
I358 K362 L372 V376 L379 E380 D538 L539 E542
Binding residue
(residue number reindexed from 1)
I54 K58 L68 V72 L75 E76 D228 L229 E232
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:4mg7, PDBe:4mg7, PDBj:4mg7
PDBsum4mg7
PubMed25260197
UniProtP03372|ESR1_HUMAN Estrogen receptor (Gene Name=ESR1)

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