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Structure of PDB 5gs4 Chain A Binding Site BS01

Receptor Information
>5gs4 Chain A (length=236) Species: 9606 (Homo sapiens) [Search protein sequence] [Download receptor structure] [Download structure with residue number starting from 1] [View receptor structure]
SLALSLTADQMVSALLDAEPPILYSESEASMMGLLTNLADRELVHMINWA
KRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLD
RNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTF
LSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLIL
SHIRHMSNKGMEHLYSMKCKNVVPLYDLLLEMLDAH
Ligand information
Receptor-Ligand Complex Structure
Global viewLocal viewStructure summary

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PDB5gs4 Structural Basis of Inhibition of ER alpha-Coactivator Interaction by High-Affinity N-Terminus Isoaspartic Acid Tethered Helical Peptides
Resolution2.4 Å
Binding residue
(original residue number in PDB)
I358 K362 L372 V376 E542
Binding residue
(residue number reindexed from 1)
I47 K51 L61 V65 E231
Enzymatic activity
Enzyme Commision number ?
External links
PDB RCSB:5gs4, PDBe:5gs4, PDBj:5gs4
PDBsum5gs4
PubMed29045135
UniProtP03372|ESR1_HUMAN Estrogen receptor (Gene Name=ESR1)

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