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Go to the GPCR, ligand, or experimental data tables.
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GPCR

Name	N-arachidonyl glycine receptor
Species	Homo sapiens (Human)
Gene	GPR18
Synonym	GPCRW G-protein coupled receptor 18 N-arachidonoyol glycine receptor NAGly receptor GPR18
Disease	N/A
Length	331
Amino acid sequence	MITLNNQDQPVPFNSSHPDEYKIAALVFYSCIFIIGLFVNITALWVFSCTTKKRTTVTIYMMNVALVDLIFIMTLPFRMFYYAKDEWPFGEYFCQILGALTVFYPSIALWLLAFISADRYMAIVQPKYAKELKNTCKAVLACVGVWIMTLTTTTPLLLLYKDPDKDSTPATCLKISDIIYLKAVNVLNLTRLTFFFLIPLFIMIGCYLVIIHNLLHGRTSKLKPKVKEKSIRIIITLLVQVLVCFMPFHICFAFLMLGTGENSYNPWGAFTTFLMNLSTCLDVILYYIVSKQFQARVISVMLYRNYLRSMRRKSFRSGSLRSLSNINSEML
UniProt	Q14330
Protein Data Bank	N/A
GPCR-HGmod model	Q14330
3D structure model	This predicted structure model is from GPCR-EXP Q14330.
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL2384898
IUPHAR	89
DrugBank	BE0002304

Ligand

Name	CHEMBL2387534
Molecular formula	C20H20O3
IUPAC name	3-benzyl-6-methoxy-5,7,8-trimethylchromen-2-one
Molecular weight	308.377
Hydrogen bond acceptor	3
Hydrogen bond donor	0
XlogP	4.9
Synonyms	BDBM50434891
Inchi Key	GWLDYBULTJKXBC-UHFFFAOYSA-N
Inchi ID	InChI=1S/C20H20O3/c1-12-13(2)19-17(14(3)18(12)22-4)11-16(20(21)23-19)10-15-8-6-5-7-9-15/h5-9,11H,10H2,1-4H3
PubChem CID	71682640
ChEMBL	CHEMBL2387534
IUPHAR	N/A
BindingDB	50434891
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Experimental Data

Parameter	Value	Reference	Database source
Activity	46.0 %	PMID23679955	ChEMBL
IC50	10000.0 nM	PMID23679955	ChEMBL

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