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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Histamine H3 receptor
Species	Mus musculus (Mouse)
Gene	Hrh3
Synonym	GPCR97 H3 receptor H3R HH3R
Disease	N/A for non-human GPCRs
Length	445
Amino acid sequence	MERAPPDGLMNASGALAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRYGVGEAGPGVETGEAGLGGGSGGGAAASPTSSSGSSSRGTERPRSLKRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGHCVPDYWYETSFWLLWANSAVNPVLYPLCHYSFRRAFTKLLCPQKLKVQPHGSLEQCWK
UniProt	P58406
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3263
IUPHAR	264
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
982	CHEMBL288431	C28H32N2O5	476.573	7 / 3	N/A	N/A
1790	ciproxifan	C16H18N2O2	270.332	3 / 1	2.5	Yes
2960	CID 44370594	C14H21N3O6	327.337	7 / 4	N/A	N/A
6499	CHEMBL128585	C17H21N3O2	299.374	3 / 2	2.7	Yes
6955	CHEMBL1641831	C19H25ClN4OS	392.946	6 / 0	4.5	Yes
9903	CHEMBL415989	C22H28N6O4	440.504	6 / 4	1.9	Yes
11131	CHEMBL181278	C27H34N2O5	466.578	6 / 1	1.6	Yes
14718	CHEMBL2436616	C31H36FN5O	513.661	6 / 1	4.4	No
16012	CHEMBL61729	C12H20N2	192.306	1 / 1	4.2	Yes
19724	CHEMBL131021	C20H24N2O6	388.42	7 / 3	N/A	N/A
19859	CHEMBL39980	C28H31NO5	461.558	6 / 2	N/A	N/A
21679	CHEMBL290613	C22H25NO6	399.443	7 / 2	N/A	N/A
24434	CHEMBL128513	C19H22N2O6	374.393	7 / 3	N/A	N/A
27740	CHEMBL35869	C24H30N2O6	442.512	8 / 2	N/A	N/A
27839	CHEMBL2436625	C28H38FN5O2	495.643	7 / 1	3.0	Yes
28412	CHEMBL39644	C23H29NO5	399.487	6 / 2	N/A	N/A
28798	CHEMBL59851	C23H23BrN2O5	487.35	6 / 3	N/A	N/A
29323	CID 44370355	C16H25N3O6	355.391	7 / 4	N/A	N/A
29722	CHEMBL2048586	C18H31N5OS	365.54	7 / 0	3.2	Yes
30344	CID 44370548	C15H23N3O7	357.363	8 / 4	N/A	N/A
30648	FUB-349	C13H16N2	200.285	1 / 1	3.2	Yes
30799	CHEMBL132798	C15H16N2O	240.306	2 / 1	3.1	Yes
32042	CHEMBL80348	C16H19N3O2	285.347	4 / 2	2.8	Yes
32405	CHEMBL277149	C14H16ClN3O2	293.751	3 / 2	2.6	Yes
33138	CHEMBL38378	C24H31NO5	413.514	6 / 2	N/A	N/A
33848	CHEMBL19172	C13H15BrN2O	295.18	2 / 1	2.8	Yes
35994	CHEMBL2436629	C25H32FN5O	437.563	6 / 1	2.2	Yes
37960	CHEMBL416053	C27H36N2O5	468.594	7 / 2	N/A	N/A
40330	CHEMBL36590	C23H29NO5	399.487	6 / 2	N/A	N/A
40692	CHEMBL303121	C15H20N2	228.339	1 / 1	4.3	Yes
41401	CHEMBL291369	C21H22N2O5	382.416	6 / 3	N/A	N/A
41862	CHEMBL560386	C23H29NO5S	431.547	6 / 0	3.7	Yes
45562	CHEMBL336499	C14H23N3O2	265.357	3 / 2	2.7	Yes
49478	CHEMBL2436617	C29H32FN5OS	517.667	7 / 1	4.6	No
50093	CHEMBL2436621	C26H31FN8O2S	538.646	9 / 1	1.5	No
50519	CHEMBL39791	C21H24FNO5	389.423	7 / 2	N/A	N/A
51535	CIPRALISANT	C14H20N2	216.328	1 / 1	3.3	Yes
52771	CID 44370617	C14H21N3O6	327.337	7 / 4	N/A	N/A
55807	CID 44351978	C17H18N2O6	346.339	7 / 3	N/A	N/A
55968	CHEMBL16593	C13H21N3O2	251.33	3 / 2	2.2	Yes
56602	Iodoproxyfan	C13H15IN2O	342.18	2 / 1	2.7	Yes
62942	CHEMBL154797	C18H29N3O6	383.445	7 / 4	N/A	N/A
62944	CHEMBL154944	C18H29N3O6	383.445	7 / 4	N/A	N/A
62948	CHEMBL155425	C18H29N3O6	383.445	7 / 4	N/A	N/A
67744	CHEMBL281187	C13H15IN2O	342.18	2 / 1	2.7	Yes
72500	CHEMBL1270264	C19H22N2O	294.398	3 / 1	3.0	Yes
72688	CHEMBL130850	C14H25N3O2	267.373	3 / 2	3.5	Yes
78373	CHEMBL335771	C12H20N2O2	224.304	3 / 1	2.6	Yes
79368	CHEMBL360791	C25H30N2O3	406.526	4 / 1	1.5	Yes
80858	CHEMBL2031602	C19H25N7S	383.518	7 / 0	3.6	Yes
83958	CHEMBL417888	C25H31NO5	425.525	6 / 2	N/A	N/A
87878	CHEMBL60342	C23H22F2N2O5	444.435	8 / 3	N/A	N/A
89009	CHEMBL129146	C22H26N2O6	414.458	7 / 3	N/A	N/A
89025	CHEMBL16592	C14H17N3O2	259.309	3 / 2	2.3	Yes
90545	CHEMBL442762	C19H22N2O7	390.392	8 / 3	N/A	N/A
90817	CID 11046028	C21H26N2O2	338.451	4 / 1	4.0	Yes
93523	CHEMBL305594	C13H14N2	198.269	1 / 1	3.0	Yes
94404	CHEMBL2048592	C22H31FN6S	430.59	8 / 0	3.9	Yes
98139	CHEMBL2048591	C22H32N6OS	428.599	8 / 1	2.8	Yes
98412	CHEMBL277989	C13H14BrN3O2	324.178	3 / 2	3.1	Yes
98897	CID 44370576	C15H23N3O6	341.364	7 / 4	N/A	N/A
99445	CHEMBL129493	C25H33N3O6	471.554	8 / 3	N/A	N/A
101313	CHEMBL419975	C12H19N3O2	237.303	3 / 2	1.6	Yes
104751	CHEMBL2048413	C17H27N5OS	349.497	6 / 0	2.4	Yes
105726	CHEMBL311828	C16H20N2O	256.349	2 / 1	3.8	Yes
106490	CHEMBL16108	C14H14F3N3O2	313.28	6 / 2	2.9	Yes
108745	CHEMBL37737	C26H33NO5	439.552	6 / 2	N/A	N/A
110195	CHEMBL1270167	C21H27NO	309.453	2 / 1	4.5	Yes
110351	CHEMBL16524	C11H17N3O2	223.276	3 / 2	1.6	Yes
111112	CHEMBL15883	C13H14N4O4	290.279	5 / 2	1.8	Yes
111434	CHEMBL128926	C23H28N2O8	460.483	9 / 3	N/A	N/A
113338	CHEMBL16274	C17H17N3O2	295.342	3 / 2	3.2	Yes
116520	CID 44370341	C16H25N3O6	355.391	7 / 4	N/A	N/A
117170	CHEMBL2375588	C21H33NO2	331.5	3 / 1	4.2	Yes
117858	CID 71458153	C15H24N2O5	312.366	6 / 3	N/A	N/A
118651	CHEMBL34844	C22H27NO5	385.46	6 / 2	N/A	N/A
119558	CHEMBL441780	C22H27NO5	385.46	6 / 2	N/A	N/A
120487	CHEMBL483400	C24H26FN3O2	407.489	5 / 0	4.0	Yes
121055	CHEMBL154478	C18H29N3O6	383.445	7 / 4	N/A	N/A
121929	CHEMBL131476	C20H27N3O2	341.455	3 / 2	4.3	Yes
123072	CHEMBL552773	C17H21ClN2O4	352.815	5 / 3	N/A	N/A
126179	CHEMBL129602	C18H19FN2O6	378.356	8 / 3	N/A	N/A
127692	CID 44370242	C17H27N3O6	369.418	7 / 4	N/A	N/A
129870	CHEMBL1270165	C20H27NO	297.442	2 / 1	4.4	Yes
132472	CHEMBL128923	C14H16N2O5	292.291	6 / 3	N/A	N/A
134868	CHEMBL2048583	C18H31N5OS	365.54	7 / 0	3.1	Yes
136010	CHEMBL495698	C26H27FN4O	430.527	5 / 0	5.0	Yes
137799	CHEMBL574387	C23H28N6OS	436.578	7 / 1	3.6	Yes
138732	CHEMBL15813	C18H24N4O2	328.416	4 / 2	2.9	Yes
139612	CHEMBL134902	C17H20N2O	268.36	2 / 1	4.1	Yes
141368	CHEMBL128357	C22H28N2O6	416.474	7 / 3	N/A	N/A
141505	CHEMBL289855	C15H22N2O3	278.352	4 / 0	3.8	Yes
144027	CHEMBL129443	C20H21N3O8	431.401	9 / 3	N/A	N/A
144457	CHEMBL279617	C13H14N4O4	290.279	5 / 2	1.8	Yes
148061	CHEMBL39705	C15H18N2O2	258.321	3 / 1	1.7	Yes
148816	CHEMBL277537	C14H16N4O4	304.306	5 / 2	1.8	Yes
150439	CHEMBL184989	C26H32N2O3	420.553	4 / 0	3.9	Yes
150454	CHEMBL130989	C20H24N2O6	388.42	7 / 3	N/A	N/A
156597	CHEMBL129403	C19H21FN2O6	392.383	8 / 3	N/A	N/A
156738	CHEMBL274262	C15H19N3O2	273.336	3 / 2	2.4	Yes

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