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GPCR

NameGrowth hormone-releasing hormone receptor
SpeciesRattus norvegicus (Rat)
GeneGhrhr
SynonymGhrfr
GHRH receptor
GRF receptor
GRFR
Growth hormone-releasing factor receptor
DiseaseN/A for non-human GPCRs
Length464
Amino acid sequenceMDSLLWATWVLCLLNLWGVALGHLHLECDFITQLRDDELACLQAAEGTNNSSMGCPGTWDGLLCWPPTGSGQWVSLPCPEFFSHFGSDPGAVKRDCTITGWSDPFPPYPVACPVPLELLTEEKSYFSTVKIIYTTGHSISIVALCVAIAILVALRRLHCPRNYIHTQLFATFILKASAVFLKDAAVFQGDSTDHCSMSTILCKVSVAVSHFATMTNFSWLLAEAVYLSCLLASTSPRSKPAFWWLVLAGWGLPVLCTGTWVGCKLAFEDTACWDLDDSSPYWWIIKGPIVLSVGVNFGLFLNIICILLRKLGPAQGGLHTRAQYCNYLLPWSCPLPQVPRERTDLGPSSHEITVQESGTRNCQLPWRLSKSTLLLIPLFGIHYIIFNFLPDSAGLGIRLPLELGLGSFQGFVVAVLYCFLNQEVRTEISRKWYGHDPELLPARRTCTEWTTPPRSRVKVLTSEC
UniProtQ02644
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL3709
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 177
Page:  / 2 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
12832D structureCHEMBL553507C31H39ClN4O4567.1275 / 4N/ANo
12842D structureCHEMBL555821C31H39ClN4O4567.1275 / 4N/ANo
65512D structureCHEMBL3301648C148H240N42O43S3327.8649 / 48-13.1No
125822D structureCHEMBL1793923C150H248N44O423339.948 / 49-12.6No
164112D structureCHEMBL1791216C148H245N43O41S3314.9148 / 48-11.7No
164122D structureCHEMBL1791236C149H247N43O41S3328.9448 / 48-11.2No
172892D structureL-692,585C32H37N7O3567.6947 / 43.8No
275212D structureCHEMBL552911C30H39N3O5521.6586 / 22.7No
275222D structureCHEMBL544536C30H39N3O5521.6586 / 22.7No
309292D structureCHEMBL553478C30H39N3O4505.6595 / 31.3No
309302D structureCHEMBL540805C30H39N3O4505.6595 / 31.3No
329992D structureBDBM50004983C143H236N40O38S3155.7645 / 47-8.5No
356972D structureCHEMBL1791192C148H244N44O41S3327.9148 / 48-12.6No
391162D structureBDBM50004968C157H261N45O43S3499.1550 / 53-10.7No
437552D structure2,4 diamino butyric acidC151H248N42O413307.947 / 47-8.2No
454282D structureCID 44387393C143H233N37O40S3142.7245 / 43-8.6No
499342D structureCHEMBL1791234C148H245N43O41S3314.9148 / 48-11.6No
500912D structureCHEMBL1791239C146H240N44O42S3315.8549 / 49-14.6No
501962D structureCHEMBL554852C32H41ClN4O4581.1545 / 4N/ANo
501972D structureCHEMBL552657C32H41ClN4O4581.1545 / 4N/ANo
530692D structureCHEMBL1791210C152H250N42O413321.9347 / 47-7.9No
530702D structureCHEMBL1791215C152H250N42O413321.9347 / 47-7.9No
530712D structureCHEMBL2369702C152H250N42O413321.9347 / 47-7.9No
568352D structureCHEMBL1791244C150H246N44O42S3369.9449 / 49-12.8No
603952D structureCHEMBL1791205C146H239N41O42S3272.8248 / 47-12.1No
631242D structureCHEMBL540800C31H42ClN3O4556.1445 / 4N/ANo
678002D structureCHEMBL1791240C147H242N44O423297.8248 / 49-13.9No
742692D structureCHEMBL1791193C146H239N43O42S3300.8448 / 48-13.0No
772272D structureCHEMBL1791242C147H242N44O42S3329.8849 / 49-14.2No
837772D structureCHEMBL553507C31H38N4O4530.6695 / 33.4No
837782D structureCHEMBL555821C31H38N4O4530.6695 / 33.4No
4450242D structureCHEMBL3348528C156H252N46O37S23428.1446 / 46-5.0No
4450252D structureCHEMBL3348527C156H252N46O37S23428.1446 / 46-5.0No
4450262D structureCHEMBL3348526C156H252N46O37S23428.1446 / 46-5.0No
4450272D structureCHEMBL3348529C156H252N46O37S23428.1446 / 46-5.0No
840662D structureCHEMBL544769C31H42ClN3O4556.1445 / 3N/ANo
840672D structureCHEMBL545465C31H42ClN3O4556.1445 / 3N/ANo
849282D structureCID 44387408C141H232N42O393139.6645 / 46-12.3No
909652D structureCHEMBL540001C28H38ClN3O2484.0813 / 3N/AN/A
917782D structureCHEMBL413900C115H187N33O312527.9636 / 36-8.0No
4454002D structureCHEMBL3350280C141H231N39O393096.6344 / 44-9.8No
929312D structureCHEMBL437650C141H231N39O393096.6344 / 44-9.8No
929322D structureCHEMBL2114075C141H231N39O393096.6344 / 44-9.8No
931432D structure91869-58-8C150H248N44O423339.948 / 52-11.3No
1031022D structureCHEMBL411774C148H240N42O43S3327.8649 / 48-13.1No
1049552D structureCHEMBL1791200C147H249N45O41S3334.9448 / 49-12.0No
1091902D structureCHEMBL1791206C146H239N41O42S3272.8248 / 47-12.1No
1117972D structureCHEMBL1791217C146H240N44O42S3315.8549 / 49-14.6No
1165852D structureCHEMBL1791203C147H243N43O41S3300.8848 / 48-12.1No
1171012D structureCID 44298521C157H253N49O41S3515.1149 / 50-9.2No
1209852D structureCHEMBL404769C148H240N42O43S3327.8649 / 48-13.7No
1229232D structureCHEMBL1791197C150H248N44O41S3355.9648 / 48-11.7No
1290692D structureCHEMBL1791209C153H252N42O413335.9547 / 47-7.5No
1303872D structureCHEMBL1791212C149H246N44O41S3341.9348 / 48-12.2No
1326382D structureCHEMBL538008C32H43N3O4533.7135 / 24.3No
1326392D structureCHEMBL545002C32H43N3O4533.7135 / 24.3No
1385902D structureCHEMBL410460C125H204N36O342755.2339 / 40-8.5No
1385912D structureCHEMBL429726C125H204N36O342755.2339 / 40-8.5No
1428072D structureCHEMBL428327C114H185N33O312513.9336 / 37-8.2No
1428082D structureCHEMBL436902C114H185N33O312513.9336 / 37-8.2No
1428092D structureCHEMBL268540C114H185N33O312513.9336 / 37-8.2No
1446152D structureCHEMBL1791202C143H242N44O41S3265.8448 / 48-14.5No
1497812D structureCHEMBL545002C32H44ClN3O4570.1715 / 3N/ANo
1497822D structureCHEMBL538008C32H44ClN3O4570.1715 / 3N/ANo
1578782D structureBDBM50004975C143H234N42O41S3229.7647 / 50-11.6No
1610382D structureCHEMBL1791228C150H248N44O42S3371.9649 / 49-12.8No
1612312D structureCHEMBL1791199C148H246N44O40S3313.9247 / 48-10.1No
1623262D structureCHEMBL427941C151H247N45O43S3412.9750 / 50-14.3No
1634222D structureCHEMBL439889C152H248N44O43S3411.9849 / 49-12.9No
1677072D structureCID 44387433C149H245N43O43S3358.9250 / 49-14.9No
1741782D structureCID 44387389C144H237N43O413226.7447 / 48-13.6No
1746682D structureBDBM50004980C144H238N42O40S3229.847 / 50-10.7No
1751272D structureCHEMBL538004C33H46ClN3O4584.1985 / 3N/ANo
1757722D structureCHEMBL265915C149H243N43O42S3340.948 / 48-12.1No
1788482D structureCHEMBL1791198C146H239N43O42S3300.8448 / 48-13.0No
1813262D structureCHEMBL429708C148H241N45O43S3370.8950 / 50-16.2No
1904012D structureCHEMBL409474C151H246N44O42S3381.9648 / 48-12.2No
1911972D structureCHEMBL1791208C151H247N45O43S3412.9750 / 50-14.9No
1916162D structureCHEMBL1791248C147H242N44O42S3329.8849 / 49-14.0No
4492692D structureCHEMBL1791233C143H242N44O42S3281.8349 / 49-14.8No
1941742D structureCID 44298170C149H244N46O39S3335.9347 / 48-11.3No
2000952D structureCHEMBL2371358C153H251N45O42S3425.0249 / 49-13.3No
2022162D structureCHEMBL1791232C147H243N43O39S3268.8846 / 46-10.4No
2026732D structureBDBM50004962C141H239N43O40S3208.7847 / 50-12.7No
2032562D structureCHEMBL1791249C146H245N45O42S3334.949 / 49-15.2No
2033542D structureCID 44298436C155H251N49O40S3473.0849 / 50-11.8No
2039142D structureCHEMBL1791225C149H246N44O41S3341.9348 / 48-12.2No
2057842D structureCHEMBL542653C27H37ClN4O5S565.1267 / 3N/ANo
2066282D structureCID 44387409C138H226N42O40S3145.6447 / 47-15.0No
2072242D structureCHEMBL1791250C146H240N44O42S3315.8549 / 49-14.6No
2075952D structureCHEMBL558422C30H37ClN4O4553.15 / 5N/ANo
2086092D structureCHEMBL1791223C148H240N42O43S3327.8649 / 48-13.7No
2173262D structureCHEMBL552657C32H40N4O4544.6965 / 33.7No
2173272D structureCHEMBL554852C32H40N4O4544.6965 / 33.7No
2183572D structureCHEMBL558422C30H36N4O4516.6425 / 40.7No
2193402D structureCHEMBL1791238C149H248N44O40S3327.9547 / 48-9.6No
2242532D structureCHEMBL544536C30H40ClN3O5558.1166 / 3N/ANo
2242542D structureCHEMBL552911C30H40ClN3O5558.1166 / 3N/ANo
2244692D structureCHEMBL1791235C151H250N44O42S3385.9949 / 49-12.3No
2290502D structureCHEMBL1791207C149H246N44O41S3341.9348 / 48-12.2No

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