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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	Adenosine receptor A1
Species	Mus musculus (Mouse)
Gene	Adora1
Synonym	A1 receptor A1-AR A1R adenosine receptor A1 RDC7
Disease	N/A for non-human GPCRs
Length	326
Amino acid sequence	MPPYISAFQAAYIGIEVLIALVSVPGNVLVIWAVKVNQALRDATFCFIVSLAVADVAVGALVIPLAILINIGPQTYFHTCLMVACPVLILTQSSILALLAIAVDRYLRVKIPLRYKTVVTQRRAAVAIAGCWILSLVVGLTPMFGWNNLSEVEQAWIANGSVGEPVIKCEFEKVISMEYMVYFNFFVWVLPPLLLMVLIYLEVFYLIRKQLNKKVSASSGDPQKYYGKELKIAKSLALILFLFALSWLPLHILNCITLFCPTCQKPSILIYIAIFLTHGNSAMNPIVYAFRIHKFRVTFLKIWNDHFRCQPKPPIEEDIPEEKADD
UniProt	Q60612
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3688
IUPHAR	18
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
1199	CHEMBL178846	C22H25ClN6O5	488.929	9 / 4	1.3	Yes
4757	CHEMBL27376	C20H20ClIN6O3	554.773	7 / 4	2.0	No
9824	CHEMBL2089350	C33H28ClN5O2	562.07	6 / 3	5.6	No
29003	CHEMBL2064639	C22H21FN6O3	436.447	8 / 4	1.1	Yes
52519	CHEMBL2402025	C29H28N6O6S	588.639	10 / 5	1.7	No
53564	CHEMBL2064655	C28H24Cl2N6O3	563.439	7 / 4	3.7	No
553500	MRS5151	C26H27ClN6O5	538.989	9 / 5	1.6	No
60679	CHEMBL2064659	C29H25ClN6O5	573.006	9 / 5	2.6	No
80517	FK-838	C21H18N4O3	374.4	5 / 1	2.1	Yes
82290	CHEMBL255907	C22H25IN6O5	580.383	9 / 4	1.0	No
90128	CHEMBL2089346	C27H25N5O2	451.53	6 / 3	3.5	Yes
92061	CHEMBL175543	C20H20Cl2N6O3	463.319	7 / 4	2.0	Yes
101162	CHEMBL283057	C14H17ClN6O3	352.779	7 / 4	-0.1	Yes
104059	CHEMBL368872	C27H27ClN6O3	519.002	7 / 4	3.3	No
446269	CHEMBL3407774	C20H20N8O3	420.433	9 / 4	-1.1	Yes
446401	CHEMBL3407783	C20H20N6O3S	424.479	8 / 4	0.7	Yes
121532	CHEMBL256520	C26H27ClN6O5	538.989	9 / 5	1.9	No
123580	CHEMBL2064656	C28H24Cl2N6O3	563.439	7 / 4	3.7	No
124376	IB-MECA	C18H19IN6O4	510.292	8 / 4	0.9	No
126973	CHEMBL425741	C20H20BrClN6O3	507.773	7 / 4	2.1	No
127343	CHEMBL2064640	C22H21ClN6O3	452.899	7 / 4	1.6	Yes
130399	CHEMBL402607	C14H17ClN6O4	368.778	8 / 4	-0.1	Yes
133231	CHEMBL2089345	C32H26ClN5O2	548.043	6 / 3	5.3	No
553964	ATL802	C24H22F3N7O3	513.481	9 / 1	2.9	No
137489	CHEMBL178644	C23H23ClN6O4	482.925	8 / 5	0.9	Yes
138949	2-Cl-IB-Meca	C18H18ClIN6O4	544.734	8 / 4	1.9	No
447755	CHEMBL3407777	C20H22N8O3	422.449	8 / 4	-0.7	Yes
165240	CHEMBL3125475	C26H28F2N2O4S	502.577	7 / 2	6.3	No
172070	CHEMBL256312	C28H33ClN8O4	581.074	9 / 6	0.7	No
182178	CHEMBL2064653	C28H25ClN6O3	528.997	7 / 4	3.1	No
188774	CHEMBL2089340	C21H20ClN5O2	409.874	6 / 3	2.6	Yes
196793	CHEMBL402574	C22H21ClN6O3	452.899	7 / 4	1.3	Yes
199445	MRS 5698	C28H23ClF2N6O3	564.978	9 / 4	3.3	No
221195	CHEMBL2064654	C28H24ClFN6O3	546.987	8 / 4	3.2	No
238312	CHEMBL2402023	C27H25N5O5S	531.587	9 / 4	2.3	No
247123	FK-453	C23H25N3O2	375.472	3 / 1	3.2	Yes
253416	CHEMBL2089335	C20H19N5O2	361.405	6 / 3	1.6	Yes
260981	Rolofylline	C20H28N4O2	356.47	3 / 1	4.9	Yes
274622	CHEMBL175444	C20H20ClIN6O3	554.773	7 / 4	1.7	No
279241	CHEMBL2064658	C28H26ClN7O3	544.012	8 / 5	2.4	No
293842	CHEMBL257405	C25H29ClN6O3Si	525.081	7 / 4	N/A	No
453338	CHEMBL3407778	C20H20N6O4	408.418	8 / 4	0.1	Yes
453818	CHEMBL3407784	C20H19ClN6O3S	458.921	8 / 4	1.7	Yes
314973	CHEMBL436649	C27H29ClN6O5	553.016	9 / 4	1.9	No
324856	CHEMBL371861	C27H22FN3O5S2	551.607	8 / 2	6.6	No
327778	CHEMBL175814	C21H23ClN6O3S	474.964	8 / 4	1.9	Yes
350087	CHEMBL411861	C22H23ClN6O3	454.915	7 / 4	1.8	Yes
351327	CHEMBL2401954	C28H25ClN6O6S	609.054	10 / 5	1.8	No
359729	CHEMBL2064661	C38H29ClN6O3	653.139	7 / 4	6.2	No
365914	CHEMBL257833	C26H27ClN6O5	538.989	9 / 5	1.6	No
375342	CHEMBL257573	C30H35ClN8O5	623.111	9 / 6	1.0	No
392276	CHEMBL2402024	C29H28N6O3	508.582	7 / 4	2.9	No
392920	CHEMBL258421	C25H27ClN6O3	494.98	7 / 4	2.8	Yes
395903	CHEMBL2064660	C34H29ClN6O3	605.095	7 / 4	4.7	No
399819	2-Chloro-N6-cyclopentyladenosine	C15H20ClN5O4	369.806	8 / 4	1.8	Yes
417310	CHEMBL257785	C28H33ClN8O4	581.074	9 / 6	0.4	No
430314	CHEMBL2401955	C28H25ClN6O6S	609.054	10 / 5	1.8	No
431160	CHEMBL2089339	C21H21N5O2	375.432	6 / 3	1.9	Yes