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GPCR

NameVasopressin V1a receptor
SpeciesMus musculus (Mouse)
GeneAvpr1a
SynonymAntidiuretic hormone receptor 1a
AVPR
AVPR V1a
AVPR1
V1A receptor
[ Show all ]
DiseaseN/A for non-human GPCRs
Length423
Amino acid sequenceMSFPRGSHDLPAGNSSPWWPLTTEGANSSREAAGLGEGGSPPGDVRNEELAKLEVTVLAVIFVVAVLGNSSVLLALHRTPRKTSRMHLFIRHLSLADLAVAFFQVLPQLCWDITYRFRGPDWLCRVVKHLQVFAMFASSYMLVVMTADRYIAVCHPLKTLQQPARRSRLMIAASWGLSFVLSIPQYFIFSVIEFEVNNGTKAQDCWATFIPPWGTRAYVTWMTSGVFVVPVIILGTCYGFICYHIWRNVRGKTASRQSKGGKGSGEAAGPFHKGLLVTPCVSSVKSISRAKIRTVKMTFVIVSAYILCWTPFFIVQMWSVWDTNFVWTDSENPSTTITALLASLNSCCNPWIYMFFSGHLLQDCVQSFPCCQSIAQKFAKDDSDSMSRRQTSYSNNRSPTNSTGTWKDSPKSSKSIRFIPVST
UniProtQ62463
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL3414410
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 18
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
4431852D structureCHEMBL3416881C25H26ClN3O3451.9513 / 03.0Yes
4437452D structureCHEMBL3416879C20H19ClN2O338.8351 / 14.4Yes
4449452D structureCHEMBL3416883C27H30ClN3O2464.0063 / 03.9Yes
4450542D structureCHEMBL3416861C21H19ClN2O2366.8452 / 13.4Yes
4463152D structureCHEMBL3416875C21H20ClN3O365.8612 / 24.1Yes
4464822D structureCHEMBL3416867C21H20N2O2332.4032 / 12.8Yes
4471492D structureCHEMBL3416872C20H18ClN3O2367.8333 / 12.4Yes
4474502D structureCHEMBL3416876C21H19ClN2O3S414.9043 / 12.9Yes
4494852D structureCHEMBL3416870C20H18ClN3O2367.8333 / 12.4Yes
4498152D structureCHEMBL3416860C29H28N2O2436.5552 / 04.7Yes
4514572D structureCHEMBL3416878C21H19ClN4O2394.8592 / 23.2Yes
4517472D structureCHEMBL3416869C27H31ClN4O3495.024 / 12.8Yes
4531582D structureCHEMBL3416868C28H31ClN4O3507.0314 / 02.8No
4532002D structureLZ0EU1YHCKC25H28ClN3O2437.9683 / 03.3Yes
4535882D structureCHEMBL3416871C20H18ClN3O2367.8333 / 12.3Yes
4569342D structureCHEMBL3416882C26H28ClN3O2449.9793 / 13.4Yes
4572382D structureCHEMBL3416884C27H30ClN3O2464.0063 / 03.8Yes
4585742D structureCHEMBL3416880C19H17Cl2N3O374.2652 / 14.4Yes

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