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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
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GPCR

Name	Gastric inhibitory polypeptide receptor
Species	Homo sapiens (Human)
Gene	GIPR
Synonym	GIP-R GIP receptor Glucose-dependent insulinotropic polypeptide receptor Gippr
Disease	Type 2 diabetes
Length	466
Amino acid sequence	MTTSPILQLLLRLSLCGLLLQRAETGSKGQTAGELYQRWERYRRECQETLAAAEPPSGLACNGSFDMYVCWDYAAPNATARASCPWYLPWHHHVAAGFVLRQCGSDGQWGLWRDHTQCENPEKNEAFLDQRLILERLQVMYTVGYSLSLATLLLALLILSLFRRLHCTRNYIHINLFTSFMLRAAAILSRDRLLPRPGPYLGDQALALWNQALAACRTAQIVTQYCVGANYTWLLVEGVYLHSLLVLVGGSEEGHFRYYLLLGWGAPALFVIPWVIVRYLYENTQCWERNEVKAIWWIIRTPILMTILINFLIFIRILGILLSKLRTRQMRCRDYRLRLARSTLTLVPLLGVHEVVFAPVTEEQARGALRFAKLGFEIFLSSFQGFLVSVLYCFINKEVQSEIRRGWHHCRLRRSLGEEQRQLPERAFRALPSGSGPGEVPTSRGLSSGTLPGPGNEASRELESYC
UniProt	P48546
Protein Data Bank	N/A
GPCR-HGmod model	P48546
3D structure model	This predicted structure model is from GPCR-EXP P48546.
BioLiP	N/A
Therapeutic Target Database	T41750
ChEMBL	CHEMBL4383
IUPHAR	248
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
7495	CHEMBL447742	C34H41N3O5	571.718	5 / 4	6.6	No
9695	CHEMBL504245	C32H31F3N4O5	608.618	9 / 4	5.5	No
11362	CHEMBL1643957	C25H24F3N7O2	511.509	9 / 2	5.5	No
13788	CHEMBL1644176	C25H24F3N7O2	511.509	9 / 2	5.9	No
25728	aminothiazole, 24	C33H26ClN3O3S	580.099	6 / 2	7.2	No
29016	aminothiazole, 4	C33H30F3N3O3S	605.676	9 / 2	7.5	No
29359	aminothiazole, 22	C30H26F3N3O5S	597.609	11 / 3	6.4	No
36907	GRA EX-25	C29H36F3N3O5	563.618	8 / 3	5.8	No
42606	CHEMBL486650	C29H30F3N3O6	573.569	9 / 4	5.2	No
50147	643011-22-7	C27H21ClF3N3O3S	559.988	9 / 2	6.4	No
50287	aminothiazole, 26	C34H26F3N3O4S	629.654	10 / 2	7.7	No
57158	CHEMBL1644198	C35H29ClF3N3O4	648.079	8 / 2	8.0	No
63643	CHEMBL217053	C18H13BrN2O4	401.216	5 / 1	3.5	Yes
64644	MK 0893	C32H27Cl2N3O4	588.485	5 / 2	6.8	No
66818	thiazole, 29	C28H22ClF3N2O4S	574.999	9 / 2	6.9	No
66986	aminothiazole, 23	C30H26F3N3O4S	581.61	10 / 3	6.1	No
471858	CHEMBL3616588	C36H31F6N3O5	699.65	12 / 2	8.6	No
75421	aminothiazole, 13	C32H29F6N3O3S	649.652	12 / 2	8.2	No
84903	CHEMBL577345	C76H95FN14O19	1527.67	22 / 18	-0.9	No
445115	GSK137647A	C16H19NO3S	305.392	4 / 1	3.5	Yes
86579	aminothiazole, 5	C38H34ClN3O3S	648.218	6 / 2	8.9	No
88004	CHEMBL198387	C29H34F3N7O3	585.632	9 / 2	5.9	No
94131	CHEMBL1644174	C25H24F3N7O2	511.509	9 / 2	5.9	No
97505	CHEMBL452310	C31H31Cl2N3O5	596.505	5 / 3	5.9	No
98585	aminothiazole, 25	C34H26F3N3O3S	613.655	9 / 2	7.4	No
99548	CHEMBL2159331	C31H22Cl2F3N3O4	628.429	8 / 2	7.6	No
109609	CHEMBL1644182	C25H16Cl2F3N7O2	574.345	9 / 2	6.3	No
115005	CHEMBL2159342	C34H31Cl2N3O3	600.54	4 / 2	8.0	No
115015	aminothiazole, 10	C30H27Cl2N3O3S	580.524	6 / 2	7.5	No
122095	CHEMBL1644185	C27H20Cl2F3N3O5	594.368	9 / 3	5.8	No
122156	CHEMBL1644189	C27H19F6N3O5	579.455	12 / 2	6.4	No
122467	CHEMBL1644199	C33H25ClF3N7O2	644.055	9 / 2	7.9	No
129592	CHEMBL2159340	C31H24Cl3N3O3	592.901	4 / 2	7.5	No
132426	CHEMBL1644183	C27H20Cl2F3N3O4	578.369	8 / 2	6.4	No
139133	CHEMBL1644184	C25H16Cl2F3N7O2	574.345	9 / 2	6.3	No
141231	CHEMBL2159343	C33H29Cl2N3O4	602.512	5 / 2	7.2	No
447299	CHEMBL1644196	C29H25ClF3N3O4	571.981	8 / 2	6.4	No
152913	CHEMBL509710	C32H32F3N3O6	611.618	9 / 4	5.0	No
153565	CHEMBL1644194	C28H24F3N3O6S	587.57	10 / 2	4.3	No
159592	thiazole, 28	C28H22ClF3N2O4S	574.999	9 / 2	6.9	No
162559	CHEMBL1644180	C26H17F6N7O3	589.458	13 / 2	6.2	No
163992	CHEMBL1933363	C24H25F3N4O3	474.484	8 / 3	4.3	Yes
173683	CHEMBL2159341	C32H27Cl2N3O3	572.486	4 / 2	7.2	No
174427	aminothiazole, 16	C27H21ClF3N3O3S	559.988	9 / 2	6.4	No
174535	CHEMBL456738	C32H34F3N3O6	613.634	9 / 4	5.8	No
192421	CHEMBL1922839	C31H33F3N8O2	606.654	9 / 2	6.4	No
192613	CHEMBL1644190	C29H23F6N3O5	607.509	12 / 2	6.6	No
192740	CHEMBL1644197	C27H21ClF3N7O2	567.957	9 / 2	6.3	No
202580	aminothiazole, 9	C29H25Cl2N3O3S	566.497	6 / 2	7.0	No
207562	CHEMBL1644203	C29H23F6N3O5	607.509	12 / 2	6.6	No
212468	CHEMBL487668	C30H31Cl2N3O5	584.494	5 / 4	6.2	No
217054	thiazole, 27	C28H22ClF3N2O3S	559.0	8 / 2	6.6	No
217108	CHEMBL452451	C32H32F3N3O8S	675.676	11 / 4	4.5	No
217616	aminothiazole, 12	C31H30F3N3O3S	581.654	9 / 2	7.3	No
219891	CHEMBL1644186	C26H18Cl2F3N7O2	588.372	9 / 2	5.9	No
221214	CHEMBL1644201	C26H17F6N7O3	589.458	13 / 2	6.2	No
222924	thiazole, 30	C29H22F6N2O5S	624.554	13 / 3	6.6	No
226823	CHEMBL1644192	C28H24F3N3O6S	587.57	10 / 2	4.3	No
227387	CHEMBL1922933	C33H32ClF3N2O4	613.074	7 / 2	8.4	No
229803	CHEMBL2159350	C33H30ClN3O5	584.069	6 / 2	6.1	No
237218	CHEMBL445532	C31H29BrF3N3O5	660.488	8 / 4	5.7	No
243031	CHEMBL1644202	C27H19F6N3O5	579.455	12 / 2	6.4	No
249761	CHEMBL1922835	C27H24ClF3N8O3	600.987	10 / 2	5.7	No
250421	CHEMBL1644200	C28H21F6N3O5	593.482	12 / 2	6.3	No
250998	aminothiazole, 3	C33H30F3N3O4S	621.675	10 / 2	7.8	No
263504	CHEMBL2159347	C32H27Cl2N3O4	588.485	5 / 2	6.8	No
265318	CHEMBL1644181	C27H20Cl2F3N3O4	578.369	8 / 2	6.4	No
268828	CHEMBL1922842	C28H24F6N8O2	618.544	12 / 2	5.6	No
273238	CHEMBL1643953	C27H28F3N3O4	515.533	8 / 2	5.6	No
277944	CHEMBL1643954	C25H24F3N7O2	511.509	9 / 2	5.6	No
278809	CHEMBL2159349	C33H27ClF3N3O4	622.041	8 / 2	7.1	No
279596	CHEMBL452311	C30H32BrN3O5	594.506	5 / 4	5.6	No
280940	CHEMBL2159338	C32H24Cl2F3N3O4	642.456	8 / 2	8.0	No
280942	CHEMBL2159337	C32H24Cl2F3N3O4	642.456	8 / 2	8.0	No
282190	CHEMBL2159339	C32H24Cl2F3N3O3	626.457	7 / 2	7.7	No
284559	CHEMBL1644191	C29H23F6N3O5	607.509	12 / 1	6.5	No
294128	CHEMBL453457	C31H32F3N3O5S	615.668	9 / 4	6.6	No
295090	aminothiazole, 15	C30H27Cl2N3O3S	580.524	6 / 2	6.9	No
295285	CHEMBL1644173	C27H28F3N3O4	515.533	8 / 2	6.0	No
298129	CHEMBL2159352	C34H30F3N3O4	601.626	8 / 2	6.8	No
298464	CHEMBL2159327	C29H26Cl3N3O4	586.894	5 / 2	6.7	No
303914	CHEMBL1933360	C24H24F3N3O4	475.468	8 / 2	4.3	Yes
310124	CHEMBL1644187	C29H23F6N3O5	607.509	12 / 2	6.7	No
313937	aminothiazole, 11	C31H28F3N3O3S	579.638	9 / 2	7.2	No
317652	aminothiazole, 1	C32H31N3O3S	537.678	6 / 2	6.6	No
318005	CHEMBL2159351	C35H34ClN3O5	612.123	6 / 2	7.0	No
320376	CHEMBL455214	C32H29F4N3O7	643.592	11 / 4	5.1	No
322388	CHEMBL1644193	C26H20F3N7O4S	583.546	11 / 2	4.3	No
324257	aminothiazole, 6	C34H26F3N3O4S	629.654	10 / 2	7.7	No
324903	aminothiazole, 20	C28H24F3N3O4S2	587.632	11 / 2	6.6	No
326616	CHEMBL528775	C31H35N3O5S	561.697	6 / 4	5.4	No
333831	CHEMBL1644188	C27H19F6N7O3	603.485	13 / 2	6.6	No
334004	CHEMBL1922840	C28H24F6N8O2	618.544	12 / 2	5.6	No
334644	CHEMBL1922834	C28H24F6N8O3	634.543	13 / 2	5.9	No
348201	CHEMBL2159353	C33H27F4N3O4	605.59	9 / 2	6.5	No
352496	aminothiazole, 19	C28H21F6N3O4S	609.543	13 / 2	7.0	No
353247	CHEMBL1933365	C26H27F3N4O3	500.522	8 / 3	4.9	No
353398	CHEMBL2159335	C30H28Cl3N3O4	600.921	5 / 2	7.1	No
355583	CHEMBL386446	C30H29Cl2N3O4	566.479	4 / 3	5.9	No
355930	CHEMBL1922841	C28H24F6N8O3	634.543	13 / 2	5.9	No