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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameProkineticin receptor 1
SpeciesHomo sapiens (Human)
GenePROKR1
SynonymVEGFR-1
PKR1
PK-R1
GPR73a
GPR73
[ Show all ]
DiseaseN/A
Length393
Amino acid sequenceMETTMGFMDDNATNTSTSFLSVLNPHGAHATSFPFNFSYSDYDMPLDEDEDVTNSRTFFAAKIVIGMALVGIMLVCGIGNFIFIAALVRYKKLRNLTNLLIANLAISDFLVAIVCCPFEMDYYVVRQLSWEHGHVLCTSVNYLRTVSLYVSTNALLAIAIDRYLAIVHPLRPRMKCQTATGLIALVWTVSILIAIPSAYFTTETVLVIVKSQEKIFCGQIWPVDQQLYYKSYFLFIFGIEFVGPVVTMTLCYARISRELWFKAVPGFQTEQIRKRLRCRRKTVLVLMCILTAYVLCWAPFYGFTIVRDFFPTVFVKEKHYLTAFYIVECIAMSNSMINTLCFVTVKNDTVKYFKKIMLLHWKASYNGGKSSADLDLKTIGMPATEEVDCIRLK
UniProtQ8TCW9
Protein Data BankN/A
GPCR-HGmod modelQ8TCW9
3D structure modelThis predicted structure model is from GPCR-EXP Q8TCW9.
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL5649
IUPHAR335
DrugBankN/A

Known ligands

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Total entries: 167
Page:  / 2 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
5361032D structureCHEMBL3938854C18H22ClN3O2S379.9034 / 13.7Yes
5339332D structureCHEMBL3983601C17H23ClN4O2S382.9075 / 13.0Yes
5361182D structureCHEMBL3941024C19H22ClN3O4S423.9126 / 12.7Yes
78792D structureCHEMBL557700C23H27Cl2N7O3520.4154 / 32.8No
4640042D structureCHEMBL3622088C20H23N5O349.4384 / 22.4Yes
5532982D structureN-{2-Furan-2-yl-1-[(pyridin-3-ylmethyl)-carbamoyl]-vinyl}-benzamideC20H17N3O3347.3744 / 22.2Yes
5339562D structureCHEMBL3901692C16H19Cl2N3O3S404.3065 / 13.6Yes
5339572D structureCHEMBL3924529C17H21ClFN3O2S385.8825 / 13.6Yes
5339622D structureCHEMBL3975166C21H25N3O3S399.5095 / 03.7Yes
5339762D structureCHEMBL3944037C20H23N3O3S385.4825 / 13.6Yes
5364352D structureCHEMBL3900231C19H23ClFN3O2S411.925 / 13.8Yes
5339772D structureCHEMBL3973527C18H23ClFN3O2S399.9095 / 03.6Yes
5364502D structureCHEMBL3987113C19H26ClN3O3S411.9455 / 13.1Yes
210952D structureCHEMBL560451C19H27Cl2N7O2456.3723 / 32.8Yes
4656582D structureCHEMBL3622087C22H28N4O364.4932 / 03.0Yes
5340062D structureCHEMBL3894644C18H24Cl2N4O2S431.3765 / 03.8Yes
256852D structureCHEMBL565054C22H27N7O4453.5035 / 30.7Yes
5340182D structureCHEMBL3966784C17H21Cl2N3O2S402.3344 / 04.1Yes
5367422D structureCHEMBL3941566C18H21ClFN3O2S397.8935 / 03.2Yes
5340242D structureCHEMBL3920852C18H24FN3O4S397.4657 / 02.5Yes
5340452D structureCHEMBL3958623C18H23ClFN3O3S415.9086 / 13.4Yes
5340472D structureCHEMBL3985917C16H19Cl2N3O3S404.3065 / 03.6Yes
5340542D structureCHEMBL3898520C19H25ClFN3O3S429.9356 / 03.5Yes
4680832D structureCHEMBL3622086C23H29N5O391.5194 / 03.3Yes
5341052D structureCHEMBL3981546C17H21Cl2N3O3S418.3335 / 23.1Yes
5341062D structureCHEMBL3946318C17H21Cl2N3O3S418.3335 / 03.7Yes
5341262D structureCHEMBL3981069C18H20Cl2N4O2S427.3445 / 13.4Yes
5341322D structureCHEMBL3897887C18H24ClN3O4S413.9176 / 03.0Yes
501402D structureCHEMBL563069C20H22ClN7O2427.8933 / 31.3Yes
4704262D structureCHEMBL3622089C20H24ClN5O385.8963 / 13.2Yes
5341842D structureCHEMBL3943549C18H21ClN4O2S392.9025 / 12.8Yes
5342032D structureCHEMBL3932513C16H19Cl2N3O3S404.3065 / 13.6Yes
5342102D structureCHEMBL3977298C16H21ClN4O2S368.885 / 23.0Yes
5342432D structureCHEMBL3986936C17H22Cl2N4O2S417.3495 / 13.7Yes
5342532D structureCHEMBL3900223C18H25N3O3S363.4765 / 13.1Yes
5342552D structureCHEMBL3973051C21H28BrN3O4S498.4366 / 03.4Yes
790502D structuretriazine compound PC1C23H29N7O3451.5314 / 31.5Yes
5379342D structureCHEMBL3927248C18H25N3O3S363.4765 / 12.3Yes
5342612D structureCHEMBL3983167C18H22F3N3O3S417.4478 / 03.3Yes
5379702D structureCHEMBL3889670C18H19ClN4O2S390.8865 / 12.6Yes
5342642D structureCHEMBL3984251C18H21ClF3N3O3S451.8898 / 03.9Yes
5381352D structureCHEMBL3905529C18H24ClN3O3S397.9185 / 22.6Yes
953132D structureCHEMBL550034C22H33N7O4459.5515 / 30.6Yes
5384292D structureCHEMBL3982097C17H21ClFN3O2S385.8825 / 13.4Yes
5343902D structureCHEMBL3980507C17H21ClFN3O2S385.8825 / 13.6Yes
5386372D structureCHEMBL3981959C17H18Cl2FN3O2S418.3085 / 13.6Yes
5343972D structureCHEMBL3910847C17H19ClF3N3O3S437.8628 / 13.9Yes
5387832D structureCHEMBL3974875C17H22ClN3O3S383.8915 / 22.4Yes
5344172D structureCHEMBL3908365C18H21Cl2N3O3S430.3445 / 03.3Yes
5387992D structureCHEMBL3893095C19H26ClN3O3S411.9455 / 02.9Yes
5344182D structureCHEMBL3956849C19H26ClN3O3S411.9455 / 03.5Yes
5388332D structureCHEMBL3917980C20H23ClN4O2S418.945 / 13.4Yes
5344352D structureCHEMBL3959736C16H21ClN4O4S400.8787 / 12.2Yes
5344362D structureCHEMBL3943716C16H19Cl2N3O3S404.3065 / 03.3Yes
5390102D structureCHEMBL3919323C17H19ClFN3O2S383.8665 / 12.9Yes
5344452D structureCHEMBL3981081C18H22F3N3O4S433.4469 / 03.6Yes
1241872D structureCHEMBL551383C21H24ClN7O3457.9194 / 31.3Yes
5344512D structureCHEMBL3912835C17H22ClN3O3S383.8915 / 03.3Yes
5344552D structureCHEMBL3926322C17H22FN3O4S383.4387 / 12.5Yes
5344582D structureCHEMBL3905662C17H23ClN4O4S414.9057 / 02.3Yes
5344622D structureCHEMBL3942364C17H21F2N3O4S401.4298 / 12.6Yes
5344732D structureCHEMBL3974638C16H20ClN3O3S369.8645 / 02.9Yes
5344852D structureCHEMBL3975181C18H22N4O3S374.4596 / 02.1Yes
5344992D structureCHEMBL3956657C18H23Cl2N3O3S432.365 / 13.1Yes
5345112D structureCHEMBL3967729C21H28ClN3O4S453.9826 / 03.3Yes
1375132D structuretriazine compound PC7C21H24FN7O3441.4675 / 30.8Yes
5345192D structureCHEMBL3917467C18H23F2N3O4S415.4568 / 02.6Yes
1395202D structureCHEMBL459142C25H31N7O3477.5694 / 31.9Yes
5345272D structureCHEMBL3938627C16H19ClFN3O3S387.8546 / 13.1Yes
1445322D structureCHEMBL560171C23H29N7O4467.535 / 31.1Yes
5345712D structureCHEMBL3889563C18H24ClN3O4S413.9176 / 22.4Yes
5400842D structureCHEMBL3898347C20H21FN4O2S400.4726 / 12.6Yes
5346422D structureCHEMBL3945817C19H27N3O3S377.5035 / 03.1Yes
5346492D structureCHEMBL3959797C17H22FN3O3S367.4396 / 02.5Yes
5346562D structureCHEMBL3955663C19H26ClN3O2S395.9464 / 14.4Yes
5346582D structureCHEMBL3963619C18H25ClN4O2S396.9345 / 03.2Yes
5346802D structureCHEMBL3895489C17H22ClN3O2S367.8924 / 13.5Yes
4840382D structureCHEMBL3622090C18H20ClFN4O362.8335 / 12.8Yes
5541392D structureIS20C23H21N3O3387.4394 / 23.1Yes
5346842D structureCHEMBL3895674C20H28ClN3O4S441.9716 / 03.0Yes
1739062D structureCHEMBL564734C21H25N7O4439.4765 / 40.3Yes
5404822D structureCHEMBL3935247C18H24ClN3O3S397.9185 / 03.5Yes
5346902D structureCHEMBL3974465C17H19ClF3N3O3S437.8628 / 03.6Yes
5405182D structureCHEMBL3953005C19H19F3N4O3S440.4419 / 13.1Yes
5405292D structureCHEMBL3949632C18H22ClF2N3O2S417.96 / 14.1Yes
5347622D structureCHEMBL3964334C18H23Cl2N3O2S416.3614 / 04.1Yes
5347712D structureCHEMBL3448261C16H20FN3O3S353.4126 / 12.5Yes
5347872D structureCHEMBL3976696C17H19ClN4O3S394.8746 / 12.7Yes
5411782D structureCHEMBL3973243C17H18Cl2FN3O2S418.3085 / 13.6Yes
2032572D structureCHEMBL563890C17H18ClN7O3403.8274 / 30.5Yes
2067262D structureCHEMBL561309C18H27N7O3389.464 / 30.4Yes
5348332D structureCHEMBL3919321C17H21BrFN3O3S446.3356 / 03.2Yes
5416552D structureCHEMBL3899695C18H24ClN3O3S397.9185 / 03.5Yes
5417192D structureCHEMBL3906648C19H26ClN3O3S411.9455 / 13.3Yes
5348782D structureCHEMBL3912045C17H20ClF2N3O3S419.8727 / 03.2Yes
2210522D structureCHEMBL552457C22H27N7O4453.5035 / 30.7Yes
5349172D structureCHEMBL3964020C17H18Cl2F3N3O3S472.3048 / 04.2Yes
5420832D structureCHEMBL3893804C17H19ClFN3O2S383.8665 / 13.1Yes
5424652D structureCHEMBL3937917C18H24ClN3O2S381.9194 / 13.8Yes
2454102D structureCHEMBL556890C18H21N7O4399.4115 / 30.1Yes

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